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Name:Tyr-(D-Dab ,Arg ,D-Trp )-cyclo-Somatostatin-14 (4-11)
Catalog No.:A0022
Structure:
Chemical Properties Cas No.:496849-46-8 Purity Limit: Synonyms:H-Tyr-cyclo(-D-Dab-Arg-Phe-Phe-D-Trp-Lys-Thr-Phe)Trifluoroacetate salt Molecular Weight:1276.51 Formula:C67H85N15O11 Storage: Solubility:
Shipping Condition
Quality Control & MSDS
Description High affinity ligand for all five somatostatin receptors (sst1-sst5). In AtT-20 mouse anterior pituitary tumor cells which mainly express sst2 and sst5 receptors the binding affinity of this somatostatin analog was found to be higher than that of somatostatin-14 (H-1490) and octreotide (H-5972). In a model of epileptogenesis, however, KE 108 did not exhibit antiepileptic activity suggesting that the high potency and efficacy of a synthetic ligand to all known somatostatin receptors may not reproduce entirely the effects of the natural ligand
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